Search results for "molecular electron density theory"

showing 10 items of 19 documents

Applications of the Conceptual Density Functional Theory Indices to Organic Chemistry Reactivity.

2016

Indexación: Web of Science Theoretical reactivity indices based on the conceptual Density Functional Theory (DFT) have become a powerful tool for the semiquantitative study of organic reactivity. A large number of reactivity indices have been proposed in the literature. Herein, global quantities like the electronic chemical potential μ, the electrophilicity ω and the nucleophilicity N indices, and local condensed indices like the electrophilic and nucleophilic Parr functions, as the most relevant indices for the study of organic reactivity, are discussed. http://www.mdpi.com/1420-3049/21/6/748

Chemical PhenomenaNucleophilicityChemistry OrganicPharmaceutical ScienceElectronsnucleophilicityReview010402 general chemistry01 natural sciencesreactivity indicesAnalytical ChemistryMolecular electron density theorylcsh:QD241-441Reactivity indicesNucleophilelcsh:Organic chemistryconceptual DFTParr functionsComputational chemistryDrug DiscoveryOrganic chemistryReactivity (chemistry)Physical and Theoretical ChemistryElectrophilicity010405 organic chemistryChemistryOrganic Chemistrymolecular electron density theory0104 chemical sciencesChemistry (miscellaneous)Conceptual DFTElectrophileMolecular MedicineQuantum TheoryDensity functional theoryelectrophilicityMolecules (Basel, Switzerland)
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Understanding the Origin of the Regioselectivity in Non-polar [3+2] Cycloaddition Reactions through the Molecular Electron Density Theory

2020

The regioselectivity in non-polar [3+2] cycloaddition (32CA) reactions has been studied within the Molecular Electron Density Theory (MEDT) at the B3LYP/6-311G(d,p) level. To this end, the 32CA reactions of nine simplest three-atom-components (TACs) with 2-methylpropene were selected. The electronic structure of the reagents has been characterized through the Electron Localisation Function (ELF) and the Conceptual DFT. The energy profiles of the two regioisomeric reaction paths and ELF topology of the transition state structures are studied to understand the origin of the regioselectivity in these 32CA reactions. This MEDT study permits to conclude that the least electronegative X1 end atom…

Electron density010405 organic chemistryChemistrymolecular electron density theoryRegioselectivityElectronic structure010402 general chemistryelectronegativity7. Clean energy01 natural sciencesCycloaddition3. Good health0104 chemical sciencesElectronegativitynon-polar [3+2] cycloaddition reactionsComputational chemistryregioselectivityAtomSingle bondNon polarmolecular mechanismorganic_chemistryTopology (chemistry)Organics
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The structural aspects of the transformation of 3-nitroisoxazoline-2-oxide to 1-aza-2,8-dioxabicyclo[3.3.0]octane derivatives: Experimental and MEDT …

2019

Abstract Reaction of 3-nitroisoxazoline-2-oxide with monosubstituted ethenes, first time documented fifty years ago, have been reviewed. Structures of phenyl and cyano derivatives of 1-aza-2,8-dioxabicyclo[3.3.0]octane produced in [3 + 2] cycloaddition (32CA) between styrene and acrylonitrile with 3-nitroisoxazoline-2-oxide were determined through single crystal XRD analysis. The molecular mechanism of the title 32CA has been also analyzed within the Molecular Electron Density Theory (MEDT) based on the M06-2X(PCM)/6-311 + G(d,p) calculations.

Electron densityElectron localization functionChemistryOrganic ChemistryOxide(3+2) cycloadditionCycloadditionElectron localization functionMolecular electron density theoryAnalytical ChemistryStyreneInorganic Chemistrychemistry.chemical_compoundPhysical chemistryAcrylonitrile3-nitroisoxazoline-2-oxideSingle crystalSpectroscopyXRD analysisOctaneJournal of Molecular Structure
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Molecular Electron Density Theory: A Modern View of Reactivity in Organic Chemistry

2016

A new theory for the study of the reactivity in Organic Chemistry, named Molecular Electron Density Theory (MEDT), is proposed herein. MEDT is based on the idea that while the electron density distribution at the ground state is responsible for physical and chemical molecular properties, as proposed by the Density Functional Theory (DFT), the capability for changes in electron density is responsible for molecular reactivity. Within MEDT, the reactivity in Organic Chemistry is studied through a rigorous quantum chemical analysis of the changes of the electron density as well as the energies associated with these changes along the reaction path in order to understand experimental outcomes. St…

Electron densitymolecular mechanismsChemistry OrganicPharmaceutical ScienceElectronsElectron010402 general chemistry01 natural sciencesArticleAnalytical Chemistrylcsh:QD241-441Electron density distributionlcsh:Organic chemistryComputational chemistryDrug DiscoveryDFT reactivity indicesNon-covalent interactionsOrganic chemistryReactivity (chemistry)Physical and Theoretical Chemistryelectron densityQuantum chemicalchemistry.chemical_classification010405 organic chemistryOrganic Chemistrymolecular electron density theory0104 chemical scienceschemistrynon-covalent interactionsModels ChemicalChemistry (miscellaneous)molecular electron density theory; DFT reactivity indices; electron localisation function; non-covalent interactions; electron density; molecular mechanisms; chemical reactivityMolecular MedicineDensity functional theoryGround stateelectron localisation functionchemical reactivityMolecules; Volume 21; Issue 10; Pages: 1319
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Unveiling the Intramolecular Ionic Diels–Alder Reactions within Molecular Electron Density Theory

2021

The intramolecular ionic Diels–Alder (IIDA) reactions of two dieniminiums were studied within the Molecular Electron Density Theory (MEDT) at the ωB97XD/6-311G(d,p) computational level. Topological analysis of the electron localization function (ELF) of dieniminiums showed that their electronic structures can been seen as the sum of those of butadiene and ethaniminium. The superelectrophilic character of dieniminiums accounts for the high intramolecular global electron density transfer taking place from the diene framework to the iminium one at the transition state structures (TSs) of these IIDA reactions, which are classified as the forward electro density flux. The activation enthalpy ass…

Exergonic reaction010405 organic chemistryChemistryintramolecular ionic Diels–Alder reactionsmolecular electron density theorydieniminiumsIntermolecular forceIminiumIonic bondingGeneral Medicine010402 general chemistry01 natural sciencesElectron localization function0104 chemical sciencesGibbs free energyChemistryCrystallographysymbols.namesakeglobal electron density transferIntramolecular forcesuperelectrophilessymbolsSingle bondQD1-999Chemistry
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Unveiling the Chemistry of Higher-Order Cycloaddition Reactions within the Molecular Electron Density Theory

2022

The higher-order cycloaddition (HOCA) reaction of tropone with cyclopentadiene (Cp) has been studied within the Molecular Electron Density Theory. The Electron Localization Function (ELF) analysis of the electronic structure of tropone and Cp characterizes the structural behaviors of the two conjugated unsaturated systems, while the conceptual DFT reactivity indices classify tropone as a strong electrophile and Cp as a strong nucleophile participating in polar cycloaddition reactions of reverse electron density flux. Eight competitive reaction paths have been characterized for this cycloaddition reaction. The most favorable one allowing the formation of the formal out [6 + 4] cycloadduct ha…

General Medicinehigher-order cycloaddition reactions; molecular electron density theory; molecular mechanism; tropone; selectivityChemistry; Volume 4; Issue 3; Pages: 735-752
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Nitropyrroles, Diels-Alder reactions assisted by microwave irradiation and solvent effect. An experimental and theoretical study

2017

The behaviors of N-tosylnitropyrroles acting as electrophilic dienophiles in polar Diels-Alder reactions joint to different dienes of increeased nucleophilicity are analyzed. The reactions were developed under microwave irradiation using toluene or protic ionic liquids (PILs) as solvents and in free solvent conditions. In all the cases explored we observed good yields in short reaction times. For these reactions, the free solvent condition and the use of protic ionic liquids as solvents offer similar results. However, the free solvent conditions favor environmental sustainability. The role of PILs in these polar Diels-Alder reactions has been theoretically studied within the Molecular Elect…

MOLECULAR ELECTRON DENSITY THEORY010402 general chemistryPhotochemistrySOLVENT EFFECTS01 natural sciencesAnalytical ChemistryInorganic Chemistrychemistry.chemical_compoundNucleophileMICROWAVEPOLAR DIELS-ALDERSpectroscopyNITROPYRROLES010405 organic chemistryOtras Ciencias QuímicasOrganic ChemistryCiencias QuímicasToluene0104 chemical sciencesSolventchemistryIonic liquidElectrophilePolarSolvent effectsCIENCIAS NATURALES Y EXACTASMicrowaveJournal of Molecular Structure
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A Molecular Electron Density Theory Study of the Competitiveness of Polar Diels–Alder and Polar Alder-ene Reactions

2018

Indexación: Scopus. Funding: Ministry of Economy and Competitiveness (MINECO) of the Spanish Government, project CTQ2016-78669-P (AEI/FEDER, UE) and Fondecyt (Chile) grant 1180348. Acknowledgments: This research was supported by the Ministry of Economy and Competitiveness (MINECO) of the Spanish Government, project CTQ2016-78669-P (AEI/FEDER, UE) and Fondecyt (Chile) grant 1180348. L.R.D. thanks Fondecyt for continuous support through Cooperación Internacional. M.R.-G. also thanks MINECO for a post-doctoral contract cofinanced by the European Social Fund (BES-2014-068258). The competitiveness of the BF3 Lewis acid (LA) catalyzed polar Diels–Alder (P-DA) and polar Alder-ene (P-AE) reactions …

Models MolecularDienePharmaceutical Science01 natural sciencesAnalytical ChemistryDioxanesAlder-ene reactionschemistry.chemical_compoundComputational chemistryDrug DiscoverySingle bondLewis acids and basesBoranesLewis AcidsCycloaddition ReactionChemistryStereoisomerismPrins reactionMolecular Electron Density Theory Diels-Alder reactionsChemistry (miscellaneous)ElectrophileThermodynamicsMolecular Medicinecompetitive reactionscompetitive reactions polar reactionsAllylic rearrangementElectrons010402 general chemistryArticleCatalysislcsh:QD241-441lcsh:Organic chemistryPseudocyclic selectivityFormaldehydeButadienespolar reactionsPhysical and Theoretical ChemistryEne reactionDiels-Alder reactionsPrins reaction pseudocyclic selectivity010405 organic chemistryOrganic ChemistryMolecular Electron Density TheoryPolar reactionsPhenanthrenespseudocyclic selectivity0104 chemical sciencesPrins reactionQuantum TheoryCompetitive reactionsMolecules
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Unveiling the Different Chemical Reactivity of Diphenyl Nitrilimine and Phenyl Nitrile Oxide in [3+2] Cycloaddition Reactions with (R)-Carvone throug…

2020

The [3+2] cycloaddition (32CA) reactions of diphenyl nitrilimine and phenyl nitrile oxide with (R)-carvone have been studied within the Molecular Electron Density Theory (MEDT). Electron localisation function (ELF) analysis of these three-atom-components (TACs) permits its characterisation as carbenoid and zwitterionic TACs, thus having a different reactivity. The analysis of the conceptual Density Functional Theory (DFT) indices accounts for the very low polar character of these 32CA reactions, while analysis of the DFT energies accounts for the opposite chemoselectivity experimentally observed. Topological analysis of the ELF along the single bond formation makes it possible to characteri…

Models MolecularNitrilemolecular mechanismsPharmaceutical Science010402 general chemistrynitrilimines01 natural sciencesArticleAnalytical Chemistrylcsh:QD241-441chemistry.chemical_compoundlcsh:Organic chemistryComputational chemistryDrug DiscoveryNitrilesSingle bondReactivity (chemistry)Physical and Theoretical ChemistryChemoselectivityCarbenoidCycloaddition ReactionMolecular Structure010405 organic chemistryChemistryNitrilimineOrganic ChemistryBiphenyl Compoundsmolecular electron density theory[3+2] cycloadditionsCycloaddition0104 chemical sciencesChemistry (miscellaneous)chemoselectivitynitrile oxidesMolecular MedicineQuantum TheoryDensity functional theoryMolecules
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Unveiling the Lewis Acid Catalyzed Diels–Alder Reactions Through the Molecular Electron Density Theory

2020

The effects of metal-based Lewis acid (LA) catalysts on the reaction rate and regioselectivity in polar Diels&ndash

Models MolecularReaction mechanismDieneChemistry OrganicMolecular ConformationNormal DistributionPharmaceutical ScienceElectrons010402 general chemistry01 natural sciencesArticleAnalytical ChemistryCatalysisReaction ratelcsh:QD241-441chemistry.chemical_compoundNucleophilelcsh:Organic chemistryComputational chemistryDrug DiscoveryButadienesLewis acids and basesPhysical and Theoretical ChemistryLewis Acidsrelation mechanismCycloaddition Reactioncatalysis010405 organic chemistryOrganic Chemistrymolecular electron density theoryRegioselectivityLewis acid0104 chemical sciences3. Good healthchemistryChemistry (miscellaneous)ElectrophileDiels–AlderSolventsMolecular MedicineQuantum TheoryThermodynamicsMolecules
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